Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50035790
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  3nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  385nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50452603(CHEMBL2371213)
Affinity DataIC50:  500nMAssay Description:Binding potency of compound in competition with [3H]CTOP for Opioid receptor mu 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016857(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  1.05E+3nMAssay Description:Binding potency of compound in competition with [3H]CTOP for Opioid receptor mu 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016857(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  1.05E+3nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016853(2-{[10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propio...)
Affinity DataIC50:  3.61E+3nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016853(2-{[10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propio...)
Affinity DataIC50:  3.62E+3nMAssay Description:Binding potency of compound in competition with [3H]CTOP for Opioid receptor mu 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016854(2-{[10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propio...)
Affinity DataIC50:  8.40E+3nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016854(2-{[10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propio...)
Affinity DataIC50:  8.40E+3nMAssay Description:Binding potency of compound in competition with [3H]CTOP for Opioid receptor mu 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50452603(CHEMBL2371213)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016858(2-{[16-(4-Amino-benzyl)-10-(4-amino-butyl)-19-(2-a...)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50016858(2-{[16-(4-Amino-benzyl)-10-(4-amino-butyl)-19-(2-a...)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding potency of compound in competition with [3H]CTOP for Opioid receptor mu 1 tested in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed