Compile Data Set for Download or QSAR
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Found 60 Enz. Inhib. hit(s) with all data for entry = 50038239
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373490(CHEMBL405260)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373490(CHEMBL405260)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373494(CHEMBL272395)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373497(CHEMBL411437)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373497(CHEMBL411437)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373494(CHEMBL272395)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373495(CHEMBL270056)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373497(CHEMBL411437)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373495(CHEMBL270056)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373494(CHEMBL272395)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373491(CHEMBL272396)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373495(CHEMBL270056)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373491(CHEMBL272396)
Affinity DataKi:  880nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373491(CHEMBL272396)
Affinity DataKi:  930nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373490(CHEMBL405260)
Affinity DataKi:  940nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373494(CHEMBL272395)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373492(CHEMBL272602)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373498(CHEMBL405292)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373492(CHEMBL272602)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373497(CHEMBL411437)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373492(CHEMBL272602)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373497(CHEMBL411437)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373498(CHEMBL405292)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373498(CHEMBL405292)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373489(CHEMBL407818)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373494(CHEMBL272395)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373491(CHEMBL272396)
Affinity DataKi:  4.40E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373492(CHEMBL272602)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373492(CHEMBL272602)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373490(CHEMBL405260)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  5.30E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373495(CHEMBL270056)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  5.50E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373496(CHEMBL272853)
Affinity DataKi:  5.50E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373489(CHEMBL407818)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373495(CHEMBL270056)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373493(CHEMBL272873)
Affinity DataKi:  8.70E+3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373498(CHEMBL405292)
Affinity DataKi:  9.70E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373489(CHEMBL407818)
Affinity DataKi:  9.90E+3nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373490(CHEMBL405260)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373493(CHEMBL272873)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50373496(CHEMBL272853)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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