Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50038734
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377972(CHEMBL1627266)
Affinity DataIC50:  1.15E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264466(CHEMBL444948 | N-Fmoc-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Gl...)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264470(CHEMBL500357 | N-Fmoc-(S)-(alpha-Me)Adi-Leu-(3'-NH...)
Affinity DataIC50:  3.90E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264461(CHEMBL508925 | N-Fmoc-Gla-Leu-(3'-NH2-Tyr)-(alpha-...)
Affinity DataIC50:  4.40E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264462(CHEMBL445342 | N-Fmoc-Adi-Leu-(3'-CH2CH2CO2H-Tyr)-...)
Affinity DataIC50:  5.60E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264465(CHEMBL462230 | N-Fmoc-Adi-Leu-(3'-NH2-Tyr)-Ac6c-Gl...)
Affinity DataIC50:  5.80E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377973(CHEMBL1627272)
Affinity DataIC50:  8.10E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264458(CHEMBL452659 | Cyclo-[CH2-CO-Gla-Leu-(3'-NH2-Tyr)-...)
Affinity DataIC50:  9.50E+3nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264456(CHEMBL502730 | Cyclo-[CH2-CO-Adi-Leu-(3'-NH2-Tyr)-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377975(CHEMBL1627245)
Affinity DataIC50:  1.70E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377976(CHEMBL1627242)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264460(CHEMBL507364 | H-Gla-Leu-(3'-NH2-Tyr)-(alpha-Me)Gl...)
Affinity DataIC50:  1.90E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377977(CHEMBL1627260)
Affinity DataIC50:  3.05E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377974(CHEMBL1627271)
Affinity DataIC50:  3.05E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264454(CHEMBL450367 | Cyclo-[CH2-CO-Adi-Leu-Tyr-(D-(alpha...)
Affinity DataIC50:  6.05E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264452(CHEMBL455745 | Cyclo-[CH2-CO-Adi-Leu-Tyr-(alpha-Me...)
Affinity DataIC50:  6.07E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264450(CHEMBL501412 | Cyclo-[CH2-CO-Adi-Leu-Tyr-(alpha-Me...)
Affinity DataIC50:  7.00E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50377971(CHEMBL1627243)
Affinity DataIC50:  7.70E+4nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264448(CHEMBL501397 | Cyclo-[CH2-CO-Adi-Leu-Tyr-(alpha-Me...)
Affinity DataIC50:  1.08E+5nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264468(CHEMBL461032 | N-Fmoc-(S)-(alpha-Me)Adi-Leu-Tyr-Ac...)
Affinity DataIC50:  1.18E+5nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264464(CHEMBL448041 | N-Fmoc-(3'-CH2CH2CO2H-Tyr)-(alpha-M...)
Affinity DataIC50:  1.68E+5nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264463(CHEMBL489405 | H-(3'-CH2CH2CO2H-Tyr)-(alpha-Me)Glu...)
Affinity DataIC50:  2.90E+5nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264469(CHEMBL499251 | N-Fmoc-(R)-(alpha-Me)Adi-Leu-(3'-NH...)
Affinity DataIC50:  7.00E+5nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50264467(CHEMBL448312 | N-Fmoc-(R)-(alpha-Me)Adi-Leu-Tyr-Ac...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity to recombinant Grb2 SH2 domain by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed