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Found 9 Enz. Inhib. hit(s) with all data for entry = 50040019
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50:  300nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 2(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of MEK2 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387975(CHEMBL2057831)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387975(CHEMBL2057831)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM14800(2-(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-et...)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387976(CHEMBL2057832)
Affinity DataIC50:  2.31E+4nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM14800(2-(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-et...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387976(CHEMBL2057832)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed