TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 2(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of MEK2 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: 2.31E+4nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Sejong University
Curated by ChEMBL
Sejong University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair