Compile Data Set for Download or QSAR
maximum 50k data
Found 61 Enz. Inhib. hit(s) with all data for entry = 50001519
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataKi:  17nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.10E+3nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282619(CHEMBL4159902)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.40E+3nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.60E+3nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43307(4-methyl-N-(4-oxidanylnaphthalen-1-yl)benzenesulfo...)
Affinity DataIC50:  2.60E+3nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282490(CHEMBL4172065)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303931(4-(dimethylamino)naphthalen-1-ol | CHEMBL571241)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282490(CHEMBL4172065)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303931(4-(dimethylamino)naphthalen-1-ol | CHEMBL571241)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282619(CHEMBL4159902)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282619(CHEMBL4159902)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43307(4-methyl-N-(4-oxidanylnaphthalen-1-yl)benzenesulfo...)
Affinity DataIC50:  1.20E+4nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303931(4-(dimethylamino)naphthalen-1-ol | CHEMBL571241)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43307(4-methyl-N-(4-oxidanylnaphthalen-1-yl)benzenesulfo...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282492(CHEMBL4170165)
Affinity DataIC50:  5.20E+4nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282628(CHEMBL4170179)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282490(CHEMBL4172065)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  8.00E+4nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303938(4-methoxynaphthalen-1-amine | CHEMBL572058)
Affinity DataIC50:  8.90E+4nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303938(4-methoxynaphthalen-1-amine | CHEMBL572058)
Affinity DataIC50:  9.50E+4nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50425036(CHEMBL2312200)
Affinity DataIC50:  1.06E+5nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50425036(CHEMBL2312200)
Affinity DataIC50:  1.41E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282628(CHEMBL4170179)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282492(CHEMBL4170165)
Affinity DataIC50:  1.77E+5nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282489(1-Naphthylamine | CHEBI:50450 | CHEMBL57394 | Naph...)
Affinity DataIC50:  1.81E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282492(CHEMBL4170165)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50425036(CHEMBL2312200)
Affinity DataIC50:  2.21E+5nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282493(CHEMBL4163878)
Affinity DataIC50:  2.50E+5nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282628(CHEMBL4170179)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50210145(CHEMBL3884307)
Affinity DataIC50:  3.10E+5nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282493(CHEMBL4163878)
Affinity DataIC50:  3.65E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282624(CHEMBL4166714)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282622(CHEMBL4174622)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282620(CHEMBL4168293)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM26195(4-aminophenol | phenol derivative, 9)
Affinity DataIC50: >5.00E+5nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282630(CHEMBL4172575)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282491(CHEMBL4168302)
Affinity DataIC50: >5.00E+5nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM26195(4-aminophenol | phenol derivative, 9)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282494(CHEMBL4161954)
Affinity DataIC50: >5.00E+5nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282493(CHEMBL4163878)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303938(4-methoxynaphthalen-1-amine | CHEMBL572058)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM14321(Fragment 18 | quinolin-4-ol)
Affinity DataIC50: >5.00E+5nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM26195(4-aminophenol | phenol derivative, 9)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282627(CHEMBL4168076)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282625(CHEMBL4172714)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 61 total ) | Next | Last >>
Jump to: