Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50041873
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)
Affinity DataKi:  3.98nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417500(CHEMBL1287877)
Affinity DataKi:  5.01nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417503(GSK-561679 | GSK561679A | NBI-77860 | VERUCERFONT)
Affinity DataKi:  6.31nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417501(CHEMBL1287904)
Affinity DataKi:  7.94nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417502(CHEMBL1287905)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417512(CHEMBL1287878)
Affinity DataKi:  25.1nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417504(CHEMBL1287936)
Affinity DataKi:  31.6nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417506(CHEMBL1287966)
Affinity DataKi:  31.6nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417511(CHEMBL1288058)
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417510(CHEMBL1288027)
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417505(CHEMBL1287965)
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417499(CHEMBL1287848)
Affinity DataKi:  63.1nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417509(CHEMBL1288026)
Affinity DataKi:  79.4nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417507(CHEMBL1287996)
Affinity DataKi:  100nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417508(CHEMBL1287997)
Affinity DataKi:  251nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417503(GSK-561679 | GSK561679A | NBI-77860 | VERUCERFONT)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences Inc

Curated by ChEMBL
LigandPNGBDBM50417502(CHEMBL1287905)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human recombinant CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed