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Found 7 Enz. Inhib. hit(s) with all data for entry = 50003422
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470684(CHEMBL173975)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470690(CHEMBL367883)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470688(CHEMBL170751)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470685(CHEMBL557158)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470689(CHEMBL171287)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470686(CHEMBL170447)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470687(CHEMBL171707)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed