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Found 14 Enz. Inhib. hit(s) with all data for entry = 50005057
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataKi:  7.00E+4nMAssay Description:Mixed type inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate preinc...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM22369(4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofu...)
Affinity DataKi:  1.90E+5nMAssay Description:Competitive inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate prein...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25753(2-{4-[2-hydroxy-3-(propan-2-ylamino)propoxy]phenyl...)
Affinity DataKi:  1.90E+5nMAssay Description:Competitive inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate prein...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataKi:  2.30E+5nMAssay Description:Competitive inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate prein...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM26197(CHEMBL112 | N-(4-hydroxyphenyl)acetamide | Norco |...)
Affinity DataKi:  2.50E+5nMAssay Description:Competitive inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate prein...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25758(2-hydroxy-5-{1-hydroxy-2-[(4-phenylbutan-2-yl)amin...)
Affinity DataKi:  2.80E+5nMAssay Description:Competitive inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate prein...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataKi:  3.00E+5nMAssay Description:Competitive inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrate prein...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM26197(CHEMBL112 | N-(4-hydroxyphenyl)acetamide | Norco |...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataIC50:  3.15E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25758(2-hydroxy-5-{1-hydroxy-2-[(4-phenylbutan-2-yl)amin...)
Affinity DataIC50:  3.60E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25753(2-{4-[2-hydroxy-3-(propan-2-ylamino)propoxy]phenyl...)
Affinity DataIC50:  3.75E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 3(Bos mutus)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM22369(4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofu...)
Affinity DataIC50:  4.30E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article