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Found 15 Enz. Inhib. hit(s) with all data for entry = 50015778
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589492(CHEMBL5171667)
Affinity DataIC50:  270nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589504(CHEMBL5202691)
Affinity DataIC50:  420nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589500(CHEMBL5208729)
Affinity DataIC50:  500nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589503(CHEMBL5199594)
Affinity DataIC50:  810nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589498(CHEMBL5182469)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589499(CHEMBL5205906)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589497(CHEMBL5190845)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589495(CHEMBL5179470)
Affinity DataIC50:  2.09E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589494(CHEMBL5180930)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589493(CHEMBL5206672)
Affinity DataIC50:  2.98E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589496(CHEMBL5169497)
Affinity DataIC50:  4.13E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589505(CHEMBL5182483)
Affinity DataIC50:  5.13E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589502(CHEMBL5198936)
Affinity DataIC50:  5.28E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50534785(CHEMBL4444989)
Affinity DataIC50:  6.78E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50589501(CHEMBL5207795)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain (1 to 424 residues) using SNAPtide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed