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Found 27 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 11156
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595565(US11591322, Compound 21)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595575(US11591322, Compound 36)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595569(US11591322, Compound 27)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595555(US11591322, Compound 5)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595556(US11591322, Compound 6 | ethyl 2-((R)-2-(((1R,4R)-...)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595576(4-(((5′-chloro-2′-(((1R,4r)-4-(((R)-1-...)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595572((S)-1-(5-(((R)-2-(((1r,4R)-4-((5′-chloro-6-(...)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595571(US11591322, Compound 30)
Affinity DataIC50: <2.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595561(US11591322, Compound 15)
Affinity DataIC50:  3.75nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595557(US11591322, Compound 8)
Affinity DataIC50:  3.75nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM126500(US11591322, Compound NVP-2 | US8778951, 310)
Affinity DataIC50:  3.75nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595577(N-(2-(2-(((1r,4r)-4-((5′-chloro-6-(((4-cyano...)
Affinity DataIC50:  3.75nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595566((R)-1-(5-(((R)-2-(((1r,4R)-4-((5′-chloro-6-(...)
Affinity DataIC50:  3.75nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595564(US11591322, Compound 19 | tert-butyl 2-((R)-2-(((1...)
Affinity DataIC50:  3.75nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595578(N-(2-(2-(((1r,4r)-4-((5′-chloro-6-(((4-cyano...)
Affinity DataIC50:  7.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595558(2-((R)-2-(((1R,4R)-4-((5′-chloro-6-(((4-cyan...)
Affinity DataIC50:  7.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595562(US11591322, Compound 16 | isopropyl 2-((R)-2-(((1r...)
Affinity DataIC50:  7.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595573(US11591322, Compound 33)
Affinity DataIC50:  7.5nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595570((R)-1-(5-(((R)-2-(((1r,4R)-4-((5′-chloro-6-(...)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595559(US11591322, Compound 12)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595563(US11591322, Compound 18)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595553(US11591322, Compound 2)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595567(US11591322, Compound 24)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595554(4-(((2′-(((1R,4R)-4-(((R)-1-((2H-tetrazol-5-...)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595560(4-(((2′-(((1R,4R)-4-(((R)-1-(1H-tetrazol-5-y...)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595568((S)-1-(5-(((R)-2-(((1r,4R)-4-((5′-chloro-6-(...)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Algen Biotechnologies

US Patent
LigandPNGBDBM595574(4-(((5′-chloro-2′-(((1R,4r)-4-(((R)-1-...)
Affinity DataIC50: >10nMAssay Description:To each well of a 96-well plate was added 5× kinase assay buffer with 10 mM DTT (6 μL), 500 μM ATP (1 μL), 5×CDK substrate (10 μL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent