Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50012067
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50114257(7-Cyclopentanecarbonyloxy-8H-indeno[1,2-d]thiazol-...)
Affinity DataEC50:  4.50E+3nMAssay Description:Effective concentration against Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50114258(5,6,7-Trimethoxy-8H-indeno[1,2-d]thiazol-2-yl-ammo...)
Affinity DataEC50:  1.70E+4nMAssay Description:Effective concentration against Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50114262(8H-Indeno[1,2-d]thiazol-2-yl-ammonium; iodide | CH...)
Affinity DataEC50:  3.80E+4nMAssay Description:Effective concentration against Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50114260(4,5-Dihydro-naphtho[1,2-d]thiazol-2-yl-ammonium; i...)
Affinity DataEC50:  1.70E+4nMAssay Description:Effective concentration against Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50114261(6-Methoxy-8H-indeno[1,2-d]thiazol-2-yl-ammonium; i...)
Affinity DataEC50:  5.00E+4nMAssay Description:Effective concentration against Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50114259(5-Methyl-8H-indeno[1,2-d]thiazol-2-yl-ammonium; io...)
Affinity DataEC50:  4.20E+3nMAssay Description:Effective concentration against Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed