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Found 20 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50017735
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604536(CHEMBL5173673)
Affinity DataEC50:  16nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604554(CHEMBL5199782)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604538(CHEMBL5191536)
Affinity DataEC50:  250nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604539(CHEMBL5204992)
Affinity DataEC50:  370nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604540(CHEMBL5173134)
Affinity DataEC50:  380nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604541(CHEMBL5207071)
Affinity DataEC50:  580nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604542(CHEMBL5203327)
Affinity DataEC50:  710nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604543(CHEMBL5172173)
Affinity DataEC50:  800nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604544(CHEMBL5191690)
Affinity DataEC50:  940nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604545(CHEMBL5196830)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  1.56E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604546(CHEMBL5195064)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604547(CHEMBL1967191)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604548(CHEMBL5196394)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604549(CHEMBL5184438)
Affinity DataEC50:  2.55E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604550(CHEMBL5194126)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604551(CHEMBL5194570)
Affinity DataEC50:  7.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604552(CHEMBL5207420)
Affinity DataEC50:  9.10E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604553(CHEMBL5186824)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604537(CHEMBL5193822)
Affinity DataEC50:  135nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed