Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50027832
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265917(4-((4-tert-butylphenyl)ethynyl)benzoic acid | CHEM...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265918(3-(4-((4-tert-butylphenyl)ethynyl)phenyl)-1,2,4-ox...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265919(3-(3-((4-tert-butylphenyl)ethynyl)phenyl)-1,2,4-ox...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265920(4-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataEC50:  0.600nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  17nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265949(3-(3-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronapht...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  0.300nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265950(5,5,8,8-tetramethyl-N-(4-(5-oxo-4,5-dihydro-1,2,4-...)
Affinity DataEC50:  520nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265951(CHEMBL1657 | TAZAROTENE | US9963439, Tazarotene | ...)
Affinity DataEC50:  63nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50265921(3-(4-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronapht...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at human RARalpha ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed