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Found 33 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50036191
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043292((1-Benzo[b]thiophen-2-yl-cyclohexyl)-cyclopropylme...)
Affinity DataIC50:  23nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043312((1-Benzo[b]thiophen-2-yl-cyclohexyl)-cyclobutylmet...)
Affinity DataIC50:  37nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043309((1-Benzo[b]thiophen-2-yl-cyclohexyl)-diethyl-amine...)
Affinity DataIC50:  42nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043295((1-Benzo[b]thiophen-2-yl-cyclohexyl)-propyl-amine ...)
Affinity DataIC50:  57nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043316(Allyl-(1-benzo[b]thiophen-2-yl-cyclohexyl)-amine |...)
Affinity DataIC50:  57nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043303((1-Benzo[b]thiophen-2-yl-cyclohexyl)-butyl-amine |...)
Affinity DataIC50:  60nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043314(CHEMBL130224 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  63nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  82nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043296((1-Benzo[b]thiophen-2-yl-cyclohexyl)-dimethyl-amin...)
Affinity DataIC50:  84nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043296((1-Benzo[b]thiophen-2-yl-cyclohexyl)-dimethyl-amin...)
Affinity DataIC50:  84nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043310((1-Benzo[b]thiophen-2-yl-cyclohexyl)-butyl-methyl-...)
Affinity DataIC50:  161nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043299((1-Benzo[b]thiophen-2-yl-cyclohexyl)-ethyl-amine |...)
Affinity DataIC50:  165nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043297(CHEMBL133223 | N*1*-(1-Benzo[b]thiophen-2-yl-cyclo...)
Affinity DataIC50:  170nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043315((1-Benzo[b]thiophen-2-yl-cyclohexyl)-ethyl-propyl-...)
Affinity DataIC50:  207nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043313((1-Benzo[b]thiophen-2-yl-cyclohexyl)-dipropyl-amin...)
Affinity DataIC50:  220nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043305((1-Benzo[b]thiophen-2-yl-cyclohexyl)-methyl-amine ...)
Affinity DataIC50:  270nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043301(CHEMBL336154 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  328nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043301(CHEMBL336154 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  328nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043304((1-Benzo[b]thiophen-2-yl-cyclohexyl)-pentyl-amine ...)
Affinity DataIC50:  337nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043311((1-Benzo[b]thiophen-2-yl-cyclohexyl)-dibutyl-amine...)
Affinity DataIC50:  386nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50040193(1-(1-Benzo[b]thiophen-2-yl-cyclohexyl)-pyrrolidine...)
Affinity DataIC50:  684nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043302(CHEMBL130383 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  713nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043302(CHEMBL130383 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  713nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043307(CHEMBL336153 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  746nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043307(CHEMBL336153 | N-(1-Benzo[b]thiophen-2-yl-cyclohex...)
Affinity DataIC50:  746nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043306(2-Amino-N-(1-benzo[b]thiophen-2-yl-cyclohexyl)-ace...)
Affinity DataIC50:  841nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043306(2-Amino-N-(1-benzo[b]thiophen-2-yl-cyclohexyl)-ace...)
Affinity DataIC50:  841nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043293(CHEMBL336575 | N*1*-(1-Benzo[b]thiophen-2-yl-cyclo...)
Affinity DataIC50:  930nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043308(CHEMBL128887 | N-[2-(1-Benzo[b]thiophen-2-yl-cyclo...)
Affinity DataIC50:  1.48E+3nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043308(CHEMBL128887 | N-[2-(1-Benzo[b]thiophen-2-yl-cyclo...)
Affinity DataIC50:  1.48E+3nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043294((1-Benzo[b]thiophen-2-yl-cyclohexyl)-[2-(3,4-dichl...)
Affinity DataIC50: >5.00E+3nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043294((1-Benzo[b]thiophen-2-yl-cyclohexyl)-[2-(3,4-dichl...)
Affinity DataIC50: >5.00E+3nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50043300(1-(1-Benzo[b]thiophen-2-yl-cyclohexyl)-imidazolidi...)
Affinity DataIC50: >5.00E+3nMAssay Description:Tested for radioligand [3H]cocaine displacement from dopamine transporter in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed