Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50041017
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  0.631nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  4nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM22915(3-(1H-imidazol-4-yl)propylphenylmethyl ether | 5-[...)
Affinity DataKi:  20nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403581(CHEMBL291369)
Affinity DataKi:  20nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403577(CHEMBL443322)
Affinity DataKi:  25nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403575(CHEMBL59679)
Affinity DataKi:  25nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403578(CHEMBL60342)
Affinity DataKi:  25nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403580(CHEMBL62244)
Affinity DataKi:  79nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403576(CHEMBL59851)
Affinity DataKi:  126nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403582(CHEMBL60606)
Affinity DataKi:  200nMAssay Description:In vitro antagonistic activity against histamine H3-receptor in an assay with K+-evoked depolarisation-induced release of [3H]histamine of synaptosom...More data for this Ligand-Target Pair
In DepthDetails Article