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Found 14 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50047301
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158897(CHEMBL3786105)
Affinity DataIC50:  1nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158896(CHEMBL3785356)
Affinity DataIC50:  2nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158894(CHEMBL3786756)
Affinity DataIC50:  2nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158893(CHEMBL3786990)
Affinity DataIC50:  4nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158891(CHEMBL3785194)
Affinity DataIC50:  4nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158895(CHEMBL3787600)
Affinity DataIC50:  4nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158898(CHEMBL3785315)
Affinity DataIC50:  4nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158889(CHEMBL3786234)
Affinity DataIC50:  5nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158901(CHEMBL3785584)
Affinity DataIC50:  8nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158899(CHEMBL3787209)
Affinity DataIC50:  9nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158900(CHEMBL3786280)
Affinity DataIC50:  9nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158892(CHEMBL3786851)
Affinity DataIC50:  9nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158902(CHEMBL3785601)
Affinity DataIC50:  13nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158890(CHEMBL3787058)
Affinity DataIC50:  14nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed