TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 1.07E+3nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 0.440nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 0.437nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Inhibitory concentration against human PDE4A isoform using a construct representing the common region of spliced variants expressed as GST-fusion pro...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rabbit whole brain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 955nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 960nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 692nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 3.02E+3nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 186nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 275nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 275nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 275nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 980nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 155nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Competitive kinetic for human alpha thrombin inhibition Ki was determinedMore data for this Ligand-Target Pair