Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for assayid = 13 entry = 50043807
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446564(CHEMBL3109404)
Affinity DataIC50:  4.84E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using GSK3 (14 to 27) as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by rad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446566(CHEMBL3109401)
Affinity DataIC50:  7.32E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using GSK3 (14 to 27) as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by rad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446565(CHEMBL3109402)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using GSK3 (14 to 27) as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by rad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed