Compile Data Set for Download or QSAR
maximum 50k data
Found 461 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 11688
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640239(3-Ethoxy-5-{6-[2-(7-fluoro-benzo[b]thiophen-5-yl)-...)
Affinity DataIC50:  1nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640244(3-Ethoxy-5-{6-[2-(4-fluoro-benzo[b]thiophen-5-yl)-...)
Affinity DataIC50:  1nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639880(3-Ethoxy-5-{6-[2-(3-methoxy-1-methyl-naphthalen-2-...)
Affinity DataIC50:  1nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639881(5-{6-[2-(3-Cyano-1-methyl-naphthalen-2-yl)-ethylam...)
Affinity DataIC50:  1nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640236(5-{6-[2-(7-Chloro-benzo[b]thiophen-5-yl)-ethylamin...)
Affinity DataIC50:  2nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639882(3-Ethoxy-5-{6-[2-(1-fluoro-3-methoxy-naphthalen-2-...)
Affinity DataIC50:  2nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640213(5-{6-[2-(1,3-Difluoro-naphthalen-2-yl)-ethylamino]...)
Affinity DataIC50:  3nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639883(3-Ethoxy-5-{6-[2-(6-methoxy-benzo[b]thiophen-5-yl)...)
Affinity DataIC50:  3nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639884(5-[6-(2-Benzo[b]thiophen-5-yl-ethylamino)-pyrimidi...)
Affinity DataIC50:  3nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639885(5-{6-[2-(7-Cyano-2,3-dihydro-benzo[1,4]dioxin-6-yl...)
Affinity DataIC50:  4nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639886(3-Ethoxy-5-{6-[2-(1-methyl-naphthalen-2-yl)-ethyla...)
Affinity DataIC50:  5nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640268(3-Ethoxy-5-{6-[2-(7-methyl-benzo[b]thiophen-5-yl)-...)
Affinity DataIC50:  6nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640300(3-(2-Ethoxy-4-{6-[2-(3-methoxy-1-methyl-naphthalen...)
Affinity DataIC50:  6nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639887(3-Ethoxy-5-{6-[2-(6-methoxy-4-methyl-benzofuran-5-...)
Affinity DataIC50:  6nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639888(3-Ethoxy-5-{6-[2-(3-methoxy-naphthalen-2-yl)-ethyl...)
Affinity DataIC50:  6nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639889(5-[6-(2-Benzo[b]thiophen-6-yl-ethylamino)-pyrimidi...)
Affinity DataIC50:  6nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639890(3-Ethoxy-5-{6-[2-(1-fluoro-naphthalen-2-yl)-ethyla...)
Affinity DataIC50:  7nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639891(3-Ethoxy-5-{6-[2-(6-methoxy-benzofuran-5-yl)-ethyl...)
Affinity DataIC50:  7nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640225(3-(3-ethoxy-5-(6-((2-(7-fluoroquinolin-6-yl)ethyl)...)
Affinity DataIC50:  8nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639892(3-Ethoxy-5-{6-[2-(6-fluoro-benzofuran-5-yl)-ethyla...)
Affinity DataIC50:  8nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639893(3-Ethoxy-5-{6-[2-(5-methoxy-benzo[b]thiophen-6-yl)...)
Affinity DataIC50:  8nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639894(5-{6-[2-(2,3-Dihydro-benzo[b]thiophen-5-yl)-ethyla...)
Affinity DataIC50:  8nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639895(3-Ethoxy-5-{6-[2-(6-fluoro-1-methyl-1H-indol-5-yl)...)
Affinity DataIC50:  8nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639896(3-Ethoxy-5-{6-[2-(1-ethynyl-naphthalen-2-yl)-ethyl...)
Affinity DataIC50:  9nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640227(4-Ethoxy-2-{6-[2-(1-methyl-naphthalen-2-yl)-ethyla...)
Affinity DataIC50:  10nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639897(4-{6-[2-(6-Methoxy-benzo[b]thiophen-5-yl)-ethylami...)
Affinity DataIC50:  10nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640217(3-(5-(6-((2-(benzo[b]thiophen-5-yl)ethyl)amino)pyr...)
Affinity DataIC50:  11nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640253(3-Ethoxy-5-{6-[2-(7-methyl-benzo[b]thiophen-6-yl)-...)
Affinity DataIC50:  11nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639898(5-{6-[2-(4-Chloro-3-methoxy-naphthalen-2-yl)-ethyl...)
Affinity DataIC50:  11nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640220(3-(5-(6-((2-(1H-indol-6-yl)ethyl)amino)pyrimidin-4...)
Affinity DataIC50:  12nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639899(3-Ethoxy-5-{6-[2-(4-methyl-benzo[b]thiophen-5-yl)-...)
Affinity DataIC50:  12nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639900(3-Ethoxy-5-{6-[2-(8-methoxy-3,4-dihydro-2H-benzo[b...)
Affinity DataIC50:  12nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640310(5-{6-[2-(7-Difluoromethoxy-2,3-dihydro-benzo[1,4]d...)
Affinity DataIC50:  13nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639901(3-Ethoxy-5-{6-[2-(8-methyl-quinolin-7-yl)-ethylami...)
Affinity DataIC50:  13nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640221(3-(5-(6-((2-(benzo[d][1,3]dioxol-5-yl)ethyl)amino)...)
Affinity DataIC50:  14nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640226(US11839613, Example 349 | {6-[4-Ethoxy-5-(1H-tetra...)
Affinity DataIC50:  14nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640333((3-Ethoxy-5-{6-[2-(7-fluoro-benzo[b]thiophen-5-yl)...)
Affinity DataIC50:  14nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639902(3-Ethoxy-5-{6-[2-(3-ethoxy-naphthalen-2-yl)-ethyla...)
Affinity DataIC50:  14nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639903(3-Ethoxy-5-{6-[2-(1H-indol-6-yl)-ethylamino]-pyrim...)
Affinity DataIC50:  15nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640328(3-(2-ethoxy-4-{6-[2-(7- fluoro-benzo[b]thiophen-5-...)
Affinity DataIC50:  16nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639905(3-Ethoxy-5-{6-[2-(7-methoxy-2,3-dihydro-benzo[1,4]...)
Affinity DataIC50:  16nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639934(5-{6-[2-(4,5-Difluoro-7-methoxy-2-methyl-benzofura...)
Affinity DataIC50:  16nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640234((4-{6-[2-(3-Cyano-1-methyl-naphthalen-2-yl)-ethyla...)
Affinity DataIC50:  17nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639906(5-{6-[2-(3-Cyano-benzo[b]thiophen-5-yl)-ethylamino...)
Affinity DataIC50:  17nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639908(4-{6-[2-(1-Fluoro-3-methoxy-naphthalen-2-yl)-ethyl...)
Affinity DataIC50:  17nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM639909(3-Ethoxy-5-{6-[2-(7-methyl-2,3-dihydro-benzo[1,4]d...)
Affinity DataIC50:  17nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640241(4-{6-[2-(7-Fluoro-benzo[b]thiophen-5-yl)-ethylamin...)
Affinity DataIC50:  18nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640329(US11839613, Example 452 | {6-[3-Ethoxy-4-(1H-tetra...)
Affinity DataIC50:  18nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640275((2-Ethoxy-6-fluoro-4-{6-[2-(7-methoxy-5-methyl-2,3...)
Affinity DataIC50:  18nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM640282(4-{6-[2-(7-Fluoro-6-methoxy-benzo[b]thiophen-5-yl)...)
Affinity DataIC50:  18nMAssay Description:The BT549 cells (NCI/No. 0507282) are detached from culture dishes with a cell dissociation buffer (Invitrogen, 13151-014), and collected in growing ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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