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Found 4 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50010107
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50091096(5-Chloro-2-(2-dimethylaminomethyl-phenylsulfanyl)-...)
Affinity DataKi:  230nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50091098(2-(2-Dimethylaminomethyl-phenylsulfanyl)-5-trifluo...)
Affinity DataKi:  1.21E+3nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50091097(3-Amino-4-(2-dimethylaminomethyl-phenylsulfanyl)-b...)
Affinity DataKi:  1.35E+3nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50091095(2-(2-Dimethylaminomethyl-phenylsulfanyl)-5-methoxy...)
Affinity DataKi:  1.99E+3nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed