Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50036386
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50036134(32+/-82-[22-cyclopropylmethyl-2,16-dihydroxy-(2S,1...)
Affinity DataKi:  0.00500nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50036140(22-cyclopropylmethyl-2,16-dihydroxy-(2S,13R)-14-ox...)
Affinity DataKi:  0.0130nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.0300nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50036137(2-[22-cyclopropylmethyl-2,16-dihydroxy-(2S,13R)-14...)
Affinity DataKi:  0.140nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50036135(5-amino(imino)methylamino-2-[22-cyclopropylmethyl-...)
Affinity DataKi:  0.160nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50036138(5-amino-2-[22-cyclopropylmethyl-2,16-dihydroxy-(2S...)
Affinity DataKi:  0.180nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50036136(6-amino-2-[22-cyclopropylmethyl-2,16-dihydroxy-(2S...)
Affinity DataKi:  0.300nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed