Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50000835
TargetEstrogen receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50261555(CHEMBL4088694)
Affinity DataEC50:  7.40E+3nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50261554(CHEMBL4092300)
Affinity DataEC50:  1.33E+3nMAssay Description:Displacement of [3H]E2 from GST-fused ERalpha-LBD (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50261553(CHEMBL4087989)
Affinity DataEC50:  1.44E+3nMAssay Description:Agonist activity at full length ERalpha (unknown origin) expressed in human HeLa cells incubated for 24 hrs by ERE-driven luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed