Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50019810
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208057(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208038(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  1.66nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208044(1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-...)
Affinity DataKi:  2.39nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208047(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208056(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  8.84nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208034(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  9.92nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208043(1-methyl-3-(R)-[4,4-Bis-(4-fluoro-phenyl)-2-oxo-im...)
Affinity DataKi:  21.9nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208036(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  27.4nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208058(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  31.5nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208039(1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-...)
Affinity DataKi:  47.8nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208035(1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-...)
Affinity DataKi:  88.5nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208051(1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-...)
Affinity DataKi:  94.5nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208029(1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-...)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208054(1-methyl-3-(S)-(2-oxo-4,4-diphenyl-imidazolidin-1-...)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208041(1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-...)
Affinity DataKi:  268nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208050(8,8-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-...)
Affinity DataKi:  498nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208031(1-methoxyethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-...)
Affinity DataKi:  552nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208030(1,1-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-...)
Affinity DataKi:  862nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208037(1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-...)
Affinity DataKi:  884nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208046(1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208033(1-cyanomethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1...)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208045(1,1-dimethyl-4-(2-oxo-4,4-diphenyl-imidazolidin-1-...)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208053(1-benzyl-1-methyl-3-(2-oxo-4,4-diphenyl-imidazolid...)
Affinity DataKi:  2.01E+3nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed