Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50034459
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362873(CHEMBL1940587)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]arginine-vasopressin from human Vasopressin V1a receptor after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362871(CHEMBL1940588)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]arginine-vasopressin from human Vasopressin V1a receptor after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362872(CHEMBL1940586)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]arginine-vasopressin from human Vasopressin V1a receptor after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed