Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50042922
TargetBeta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50433269(CHEMBL2376303)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50433274(CHEMBL2376321)
Affinity DataIC50:  126nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50433272(CHEMBL2376325)
Affinity DataIC50:  398nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-mannosyl-glycoprotein 4-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50433273(CHEMBL2376322)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed