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Found 2 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50014626
TargetCytochrome P450 2C19(Homo sapiens (Human))
Henan Normal University

Curated by ChEMBL
LigandPNGBDBM50103597(Antra | CHEBI:77260 | H 168/68 | H-168/68 | Losec ...)
Affinity DataIC50:  2.55E+3nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate incubated for 10 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Henan Normal University

Curated by ChEMBL
LigandPNGBDBM50578131(CHEMBL4864983)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate incubated for 10 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed