Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50016748
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173091(4-(4-Chloro-phenyl)-piperazine-1-carboxylic acid [...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173098(4-(2-Methoxy-phenyl)-piperazine-1-carboxylic acid ...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173094(4-(4-Methylsulfanyl-phenyl)-piperazine-1-carboxyli...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173093(1-(2-Methoxy-phenyl)-piperidine-4-carboxylic acid ...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173090(4-(4-Fluoro-phenyl)-piperazine-1-carboxylic acid [...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173096(4-Biphenyl-4-yl-piperazine-1-carboxylic acid [4-me...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173092(4-(2-Fluoro-phenyl)-piperazine-1-carboxylic acid [...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173097(4-(4-Trifluoromethyl-phenyl)-piperazine-1-carboxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50173095(4-(2-Chloro-phenyl)-piperazine-1-carboxylic acid [...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity towards cloned Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed