Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50035521
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026972(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  226nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026973(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026969(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  730nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  1.03E+3nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026963(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  2.05E+3nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026966(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  7.70E+4nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed