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Found 2 Enz. Inhib. hit(s) with all data for assayid = 6 entry = 50001790
TargetGlucocorticoid receptor(Sus scrofa)
Oric Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at GR in mini pig PBMC assessed as reduction in dexamethasone-induced GILZ gene expression incubated for 24 hrs by RT-qPCR methodMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Sus scrofa)
Oric Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50368933(CHEMBL4161754)
Affinity DataIC50:  181nMAssay Description:Antagonist activity at GR in mini pig PBMC assessed as reduction in dexamethasone-induced GILZ gene expression incubated for 24 hrs by RT-qPCR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed