Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for assayid = 6 entry = 50002099
TargetEstrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50453439(CHEMBL4209440)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at CMV-fused ERalpha-LBD-GAL4-DBD (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50453435(CHEMBL4210210)
Affinity DataIC50:  4.10E+3nMAssay Description:Antagonist activity at CMV-fused ERalpha-LBD-GAL4-DBD (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50453447(CHEMBL4211975)
Affinity DataIC50:  4.70E+3nMAssay Description:Antagonist activity at CMV-fused ERalpha-LBD-GAL4-DBD (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50453441(CHEMBL4202476)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at CMV-fused ERalpha-LBD-GAL4-DBD (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed