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Found 46 Enz. Inhib. hit(s) with all data for assayid = 6 entry = 50048220
LigandPNGBDBM50208626(CHEMBL3884821)
Affinity DataIC50:  18nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50140932(CHEMBL3753668)
Affinity DataIC50:  21nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208635(CHEMBL3883660)
Affinity DataIC50:  25nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208625(CHEMBL3885431)
Affinity DataIC50:  27nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  29nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
LigandPNGBDBM50208729(CHEMBL3883764)
Affinity DataIC50:  50nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208715(CHEMBL3884570)
Affinity DataIC50:  180nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208627(CHEMBL3885316)
Affinity DataIC50:  200nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208639(CHEMBL3883414)
Affinity DataIC50:  310nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208709(CHEMBL3883639)
Affinity DataIC50:  370nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208638(CHEMBL3883820)
Affinity DataIC50:  370nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208633(CHEMBL3884015)
Affinity DataIC50:  440nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208710(CHEMBL3884627)
Affinity DataIC50:  600nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208636(CHEMBL3884932)
Affinity DataIC50:  600nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208637(CHEMBL3884845)
Affinity DataIC50:  670nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208724(CHEMBL3884250)
Affinity DataIC50:  850nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208711(CHEMBL3885335)
Affinity DataIC50:  850nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208716(CHEMBL3885328)
Affinity DataIC50:  870nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208624(CHEMBL3885360)
Affinity DataIC50:  970nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208630(CHEMBL3751934)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50140930(CHEMBL3753970)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208641(CHEMBL3884086)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208634(CHEMBL3884861)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208632(CHEMBL3883541)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208726(CHEMBL3885043)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208720(CHEMBL3884583)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208725(CHEMBL3883458)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208628(CHEMBL3885036)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208643(CHEMBL3885021)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208719(CHEMBL3885333)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50140923(CHEMBL3753955)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208640(CHEMBL3883448)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50140931(CHEMBL3753782)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50140929(CHEMBL3754608)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208714(CHEMBL3884031)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208631(CHEMBL3884764)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208629(CHEMBL3884241)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208723(CHEMBL3883580)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208708(CHEMBL3883813)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208713(CHEMBL3885092)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208718(CHEMBL3885482)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208728(CHEMBL3885267)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208712(CHEMBL3883356)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208642(CHEMBL3883943)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208722(CHEMBL3884113)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50208727(CHEMBL3884027)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed