Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for assayid = 7 entry = 50042783
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430963(CHEMBL2337842)
Affinity DataKi:  200nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430964(CHEMBL2337841)
Affinity DataKi:  316nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataKi:  5.03E+3nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed