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Found 2 Enz. Inhib. hit(s) with all data for assayid = 7 entry = 50047176
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inverse agonist activity at human RORgamma transfected in HEK293 cells after 24 hrs by beta galactosidase luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50152147(CHEMBL3781062)
Affinity DataIC50:  4.30E+4nMAssay Description:Inverse agonist activity at human RORgamma transfected in HEK293 cells after 24 hrs by beta galactosidase luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed