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Found 4 of ph data with Target = 'Acetylpolyamine amidohydrolase'
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University Of Pennsylvania

LigandPNGBDBM152730(7-Amino-N-hydroxypentanamide (6))
Affinity DataIC50:  68nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University Of Pennsylvania

LigandPNGBDBM152729(6-Amino-N-hydroxypentanamide (5))
Affinity DataIC50:  130nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University Of Pennsylvania

LigandPNGBDBM152731(8-Amino-N-hydroxypentanamide (7))
Affinity DataIC50:  150nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University Of Pennsylvania

LigandPNGBDBM152728(5-Amino-N-hydroxypentanamide (4))
Affinity DataIC50:  170nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed