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Found 121
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  9.5nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  26.9nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383373(CHEMBL592652 | GSK0660)
Affinity DataIC50:  48nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383370(CHEMBL2030543)
Affinity DataIC50:  52nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383370(CHEMBL2030543)
Affinity DataIC50:  180nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  370nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383372(CHEMBL1998001)
Affinity DataIC50: >500nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  610nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50508127(CHEMBL4449687)
Affinity DataIC50:  960nMAssay Description:Antagonist activity at mouse PPARdeltaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50:  1.39E+3nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50081222(2-(4-{2-[1-Cycloheptyl-3-(2,4-difluoro-phenyl)-ure...)
Affinity DataEC50:  1.40E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50081225(2-(4-{2-[3-(4-Fluoro-phenyl)-1-heptyl-ureido]-ethy...)
Affinity DataEC50:  5.50E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50081224(2-(4-{2-[1-(5-Cyclohexyl-pentyl)-3-(4-fluoro-pheny...)
Affinity DataEC50:  2.30E+4nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  1.10E+5nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50081223(2-(4-{2-[3-(2,4-Difluoro-phenyl)-1-heptyl-ureido]-...)
Affinity DataEC50:  3.20E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.60E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50085040(CHEMBL278994 | L-796449 | {3-Chloro-4-[3-(3-phenyl...)
Affinity DataEC50:  23nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50:  7.20E+3nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  1.10E+5nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28662(2-[4-(3-{[2-(2-chloro-6-fluorophenyl)ethyl][(2,3-d...)
Affinity DataEC50:  410nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  2.90E+3nMAssay Description:Activation of murine PPAR delta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  19nMAssay Description:Agonist activity against PPAR deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  30nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  20nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50176605((S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse PPARdelta transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50207469(CHEMBL222880 | {4-[3,3-bis-(4-bromo-phenyl)-allyls...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229209(CHEMBL404467 | N-(4-(4-methylphenylsulfonamido)ben...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229217(CHEMBL402100 | N-(4-(2,2,2-trifluoroacetamido)benz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229215(CHEMBL254540 | N-(4-((2H-tetrazol-5-yl)methoxy)ben...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229208(CHEMBL427890 | N-(4-(2,2,2-trifluoroethylsulfonami...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229206(CHEMBL253310 | N-(4-(trifluoromethylsulfonamido)be...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229222(CHEMBL253109 | N-(4-(butylsulfonamido)benzyl)-4-me...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229212(CHEMBL254946 | N-(4-(propan-2-ylsulfonamido)benzyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229205(CHEMBL253520 | N-(4-((trifluoromethylsulfonamido)m...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229219(4'-chloro-biphenyl-4-carboxylic acid 4-trifluorome...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229211(CHEMBL254743 | N-(4-(2-methyl-1-oxo-1-(trifluorome...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229220(CHEMBL254744 | N-(4-(methylsulfonamido)benzyl)-4-m...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50229216(CHEMBL254742 | N-(4-(2-hydroxy-3,4-dioxocyclobut-1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50246525(2-(4-((5-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at mouse PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50245782(2-(4-((5-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  7.10E+3nMAssay Description:Agonist activity at mouse PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50245843(2-(4-((5-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at mouse PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50245945(2-(4-((1-allyl-5-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at mouse PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50246088(2-methyl-2-[2-methyl-4-({[1-methyl-5-(2'-methyl-bi...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at mouse PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50306508(4'-((2,3-dimethyl-5-(1-phenylpropylcarbamoyl)-1H-i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta expressed in african green monkey CV1 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50306518(4'-((6-(1-phenylpropylcarbamoyl)-2-propyl-1H-benzo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta expressed in african green monkey CV1 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse PPARdelta expressed in african green monkey CV1 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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