Compile Data Set for Download or QSAR
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Found 4
TargetPup--protein ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM36880(2,2'-THIOBIS(4,6-DICHLOROPHENOL) | 2,4-dichlor...)
Affinity DataIC50:  1.59E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PafA expressed in Escherichia coli BL-21(DE3) assessed as inhibition of pup-ylation using Mtb PanB substrate...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPup--protein ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50124518((E)-3-(3'-Adamantan-1-yl-4'-hydroxy-biphenyl-4-yl)...)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PafA expressed in Escherichia coli BL-21(DE3) assessed as inhibition of pup-ylation using Mtb PanB substrate...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPup--protein ligase(Corynebacterium glutamicum (strain ATCC 13032 / DS...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594452(SEPANTRONIUM | Sepantronium cation | Sepantronium ...)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of Corynebacterium glutamicum PafA expressed in Escherichia coli BL-21(DE3) assessed as pup-ylation using Mtb KasA substrate by SDS-PAGE a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPup--protein ligase(Corynebacterium glutamicum (strain ATCC 13032 / DS...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594452(SEPANTRONIUM | Sepantronium cation | Sepantronium ...)
Affinity DataEC50:  1.70E+3nMAssay Description:Activation of Corynebacterium glutamicum PafA expressed in Escherichia coli BL-21(DE3) assessed as pup-ylation using Mtb PanB substrate by SDS-PAGE a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed