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Found 6
TargetPiezo-type mechanosensitive ion channel component 1(Mus musculus)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50600401(CHEMBL4303374)
Affinity DataEC50:  1.71E+4nMAssay Description:Agonist activity at mouse Piezo1 transfected in human HEK293T cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPiezo-type mechanosensitive ion channel component 1(Mus musculus)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50600401(CHEMBL4303374)
Affinity DataKd:  4.56E+4nMAssay Description:Binding affinity to CM5 sensor chip-immobilized mouse Piezo1 (1 to 2190 residues) assessed as dissociation constant by real-time SPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPiezo-type mechanosensitive ion channel component 1(Mus musculus)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50600403(CHEMBL5181053)
Affinity DataKd:  2.24E+6nMAssay Description:Binding affinity to mouse Piezo1 assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPiezo-type mechanosensitive ion channel component 1(Mus musculus)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50600403(CHEMBL5181053)
Affinity DataEC50:  1.58E+5nMAssay Description:Inhibition of mouse Piezo1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPiezo-type mechanosensitive ion channel component 1(Mus musculus)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50600402(CHEMBL5208985)
Affinity DataKd:  2.75E+6nMAssay Description:Binding affinity to mouse Piezo1 assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPiezo-type mechanosensitive ion channel component 1(Mus musculus)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50600402(CHEMBL5208985)
Affinity DataEC50:  2.00E+5nMAssay Description:Inhibition of mouse Piezo1More data for this Ligand-Target Pair
In DepthDetails PubMed