TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 940nMAssay Description:Agonist activity at GPR88 in mouse striatal membranes assessed as increase in [35S]-GTP-gammaS bindingMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 1.14E+3nMAssay Description:Agonist activity at GPR88 in wild type mouse striatal membranes assessed as increase in [35S]-GTPgammaS binding after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 535nMAssay Description:Agonist activity at GPR88 in wild type mouse striatal membranes assessed as increase in [35S]-GTPgammaS binding after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 6.50E+3nMAssay Description:Agonist activity at wild type GPR88 expressed in C57BL/6J mouse striatal membrane assessed as [35S] GTPgammaS binding incubated for 1 hr by liquid sc...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 942nMAssay Description:Agonist activity at GPR88 in mouse striatal membrane assessed as [35S]-GTPgammaS-binding by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 41nMAssay Description:Binding affinity to GPR88 in mouse striatal membrane by filtration methodMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 8.90E+3nMAssay Description:Agonist activity at wild type GPR88 expressed in mouse striatal membrane assessed as [35S] GTPgammaS binding incubated for 1 hr by liquid scintillati...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at GPR88 in mouse striatal membrane assessed as [35S]-GTPgammaS-binding by liquid scintillation countingMore data for this Ligand-Target Pair