TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 0.360nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as reduction in channel current with holding potential 0 mV and ramp voltage ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 0.380nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as reduction in channel current with holding potential 0 mV and ramp voltage ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as decrease in intracellular calcium level at membrane potential -120 mV for ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as decrease in intracellular calcium level at membrane potential -120 mV for ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as decrease in intracellular calcium level at membrane potential -120 mV for ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 2.60nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as reduction in channel current with holding potential 0 mV and ramp voltage ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 3.80nMAssay Description:Inhibition of recombinant human SK3 expressed in HEK293T cells assessed as decrease in intracellular calcium level at membrane potential -120 mV for ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Inhibition of human Kca 2.3 expressed in HEK293 cells by patch clamp techniqueMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Potentiation of human KCa2.3 expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiology relative ...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Inhibition of wild type human SK3 channel expressed in HEK293 cells assessed as Ca2+ sensitivity by inside-out patch clamp techniqueMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Potentiation of human KCa2.3 expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 1.81E+3nMAssay Description:Inhibition of wild type human SK3 channel expressed in HEK293 cells assessed as Ca2+ sensitivity by inside-out patch clamp techniqueMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Inhibition of wild type human SK3 channel expressed in HEK293 cells assessed as Ca2+ sensitivity by inside-out patch clamp technique in presence of 5...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 1.50E+4nMpH: 7.35 T: 2°CAssay Description:All experiments were conducted at room temperature (22-24° C.) with an EPC-10 amplifier and Pulse software (HEKA, Lambrecht/Pfalz, Germany) in the wh...More data for this Ligand-Target Pair