TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Partial agonist activity against homomeric rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 1.75E+4nMAssay Description:Partial agonist activity with low efficacy against rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 3.45E+4nMAssay Description:Full agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 7.00E+4nMAssay Description:Partial agonist activity againast human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 1.01E+5nMAssay Description:Activation of human rho2 GABA-C receptor at 34% of maximal GABA-induced responseMore data for this Ligand-Target Pair