Compile Data Set for Download or QSAR
maximum 50k data
Found 292 of ic50 data for polymerid = 2331
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461249(CHEMBL1215628)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461265(CHEMBL4226307)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50243232(CHEMBL486232 | GNF-PF-5434 | N-((S)-4-methyl-1-oxo...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461271(CHEMBL4224764)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461272(CHEMBL4227031)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461269(CHEMBL4227166)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033708(CHEMBL3358129)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461270(CHEMBL4227486)
Affinity DataIC50:  3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033628(CHEMBL3358142)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461267(CHEMBL4227427)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033761(CHEMBL3358128)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033625(CHEMBL3352874)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461260(CHEMBL4228926)
Affinity DataIC50:  8nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461266(CHEMBL4226577)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of FP2' in Plasmodium falciparum trophozoite stage after 1 hr by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of FP2 in Plasmodium falciparum trophozoite stage after 1 hr by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461264(CHEMBL4227848)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033630(CHEMBL3358141)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033626(CHEMBL3358144)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033627(CHEMBL3358143)
Affinity DataIC50:  12nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  15nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  15nMAssay Description:Inhibition of falcipain2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  20nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain 2 expressed in Escherichia coli using Z-Leu-Arg-AMC as substrate incubated for 30 min prior...More data for this Ligand-Target Pair
In DepthDetails Article
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataIC50:  20nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461247(CHEMBL4228861)
Affinity DataIC50:  23nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50033659(CHEMBL3358140)
Affinity DataIC50:  25nMAssay Description:Inhibition of Plasmodium falciparum FP2 using Z-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461268(CHEMBL4225350)
Affinity DataIC50:  26nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461248(CHEMBL4227295)
Affinity DataIC50:  27nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513155(CHEMBL4434685)
Affinity DataIC50:  29nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513162(CHEMBL4467013)
Affinity DataIC50:  31nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513158(CHEMBL4439637)
Affinity DataIC50:  33nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461273(CHEMBL4227696)
Affinity DataIC50:  55nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461256(CHEMBL4228143)
Affinity DataIC50:  57nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513163(CHEMBL4442854)
Affinity DataIC50:  57nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513161(CHEMBL4472824)
Affinity DataIC50:  59nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513167(CHEMBL4564002)
Affinity DataIC50:  60nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM12042((2R,3R)-3-{[(1S)-1-[(4-carbamimidamidobutyl)carbam...)
Affinity DataIC50:  68nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513156(CHEMBL4442674)
Affinity DataIC50:  84nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50258544(CHEMBL4096388)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461252(CHEMBL4224829)
Affinity DataIC50:  137nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50456905(CHEMBL2235031)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli using peptide substrate by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50456905(CHEMBL2235031)
Affinity DataIC50:  150nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain 2 expressed in Escherichia coli using Z-Leu-Arg-AMC as substrate incubated for 30 min prior...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513166(CHEMBL4527228)
Affinity DataIC50:  156nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513159(CHEMBL4516951)
Affinity DataIC50:  169nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50486819(CHEMBL2235039)
Affinity DataIC50:  170nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain 2 expressed in Escherichia coli using Z-Leu-Arg-AMC as substrate incubated for 30 min prior...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461257(CHEMBL4228343)
Affinity DataIC50:  178nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461250(CHEMBL4227965)
Affinity DataIC50:  192nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50486810(CHEMBL2235030)
Affinity DataIC50:  210nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain 2 expressed in Escherichia coli using Z-Leu-Arg-AMC as substrate incubated for 30 min prior...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461261(CHEMBL4229174)
Affinity DataIC50:  230nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50513168(CHEMBL4437416)
Affinity DataIC50:  235nMAssay Description:Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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