Compile Data Set for Download or QSAR
maximum 50k data
Found 77 of ic50 data for polymerid = 49000301
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071739((S)-3-(1H-Indol-3-yl)-N-[1-(5-methoxy-pyridin-2-yl...)
Affinity DataIC50:  0.660nMAssay Description:Antagonistic activity against labelled Bombesin receptor bb1 binding sites in rat olfactory bulb by using [125I]- [Tyr] bombesin in presence of [D-Ph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158699(CHEMBL414307 | [(N4-Bzdig)0]BB(7-14))
Affinity DataIC50:  0.900nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158702(CHEMBL413893 | Universal ligand)
Affinity DataIC50:  0.960nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158698(CHEMBL266078 | [N40,Pro1,Tyr4]BB)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158700(CHEMBL266079 | [(N4-Bzdig)0,Nle14]BB(7-14))
Affinity DataIC50:  2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158697(CHEMBL268222 | [N40,Pro1,Tyr4,Nle 14]BB)
Affinity DataIC50:  11.2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147019(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-methoxy-2,...)
Affinity DataIC50:  29nMAssay Description:Affinity of [125I][D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147019(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-methoxy-2,...)
Affinity DataIC50:  29nMAssay Description:Affinity of [125I][D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)
Affinity DataIC50:  96nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)
Affinity DataIC50:  96nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295222(10-butyl-11-(2-chloro-6-fluorophenyl)-3,3,8-trimet...)
Affinity DataIC50:  150nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295254(11-(2-chloro-6-fluorophenyl)-3,3,8,10-tetramethyl-...)
Affinity DataIC50:  170nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295221(11-(2-chloro-6-fluorophenyl)-10-ethyl-3,3,8-trimet...)
Affinity DataIC50:  180nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295245(3,3,8-trimethyl-11-(2-(methylthio)phenyl)-2,3,4,5,...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295232(11'-(2-chlorophenyl)-8'-methyl-4',5',10',11'-tetra...)
Affinity DataIC50:  240nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295233(8'-methyl-11'-(2-(methylthio)phenyl)-4',5',10',11'...)
Affinity DataIC50:  250nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295246(3,3,8-trimethyl-11-(2-(trifluoromethyl)phenyl)-2,3...)
Affinity DataIC50:  250nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295247(11-(2-chlorophenyl)-3,3,8-trimethyl-2,3,4,5,10,11-...)
Affinity DataIC50:  280nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295223(11'-(2-chloro-6-fluorophenyl)-8'-methyl-4',5',10',...)
Affinity DataIC50:  280nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295236(11-(2-chloro-6-fluorophenyl)-3,3,8-trimethyl-2,3,4...)
Affinity DataIC50:  300nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147021(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-2,3,4,9-tetr...)
Affinity DataIC50:  320nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataIC50:  350nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295237(11-(2-chloro-6-fluorophenyl)-3,3-dimethyl-8-(trifl...)
Affinity DataIC50:  370nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295224(11-(2-chloro-6-fluorophenyl)-3,8-dimethyl-2,3,4,5,...)
Affinity DataIC50:  450nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295234(11'-(2-fluoro-6-(trifluoromethyl)phenyl)-8'-methyl...)
Affinity DataIC50:  540nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295248(3,3,8-trimethyl-11-(2-nitrophenyl)-2,3,4,5,10,11-h...)
Affinity DataIC50:  550nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)
Affinity DataIC50:  580nMAssay Description:Antagonist activity at human neuromedin B receptor transfected in HEK293 cells assessed as inhibition of 1 nM neuromedin B-induced myo-[3H]inositol p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147035(3-[3-(2-Methyl-4-nitro-phenyl)-ureido]-2,3,4,9-tet...)
Affinity DataIC50:  620nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295235(8'-methyl-11'-(2-(trifluoromethylthio)phenyl)-4',5...)
Affinity DataIC50:  640nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147043(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-methyl-2,3...)
Affinity DataIC50:  660nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147036(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-4,6-dimethyl...)
Affinity DataIC50:  700nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147036(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-4,6-dimethyl...)
Affinity DataIC50:  700nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147031(3-[3-(4-Nitro-phenyl)-ureido]-2,3,4,9-tetrahydro-1...)
Affinity DataIC50:  800nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295225(11-(2-chloro-6-fluorophenyl)-3-isopropyl-8-methyl-...)
Affinity DataIC50:  810nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295238(8-chloro-11-(2-chloro-6-fluorophenyl)-3,3-dimethyl...)
Affinity DataIC50:  860nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147023(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-4,7-difluoro...)
Affinity DataIC50:  1.01E+3nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295249(11-(2-methoxyphenyl)-3,3,8-trimethyl-2,3,4,5,10,11...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147041(3-[3-(4-Trifluoromethyl-phenyl)-ureido]-2,3,4,9-te...)
Affinity DataIC50:  1.11E+3nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295250(11-(2-fluorophenyl)-3,3,8-trimethyl-2,3,4,5,10,11-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295239(11-(2-chloro-6-fluorophenyl)-3,3-dimethyl-8-(trifl...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295240(11-(2-chloro-6-fluorophenyl)-3,3-dimethyl-1-oxo-2,...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295226(11-(2-chloro-6-fluorophenyl)-8-methyl-2,3,4,5,10,1...)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147029(5-(3-{3-[(1-Pyridin-2-yl-cyclohexylmethyl)-carbamo...)
Affinity DataIC50:  1.85E+3nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147040(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-trifluorom...)
Affinity DataIC50:  1.89E+3nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295227(11-(2-chloro-6-fluorophenyl)-3-(4-methoxyphenyl)-8...)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147028(7-Bromo-3-[3-(2,6-diisopropyl-phenyl)-ureido]-2,3,...)
Affinity DataIC50:  2.14E+3nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295241(11-(2-chloro-6-fluorophenyl)-8-methoxy-3,3-dimethy...)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147020(3-[3-(3-Acetyl-phenyl)-ureido]-2,3,4,9-tetrahydro-...)
Affinity DataIC50:  2.27E+3nMAssay Description:Affinity of [125I]-[D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295251(11-(2,6-difluorophenyl)-3,3,8-trimethyl-2,3,4,5,10...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295228(11-(2-chloro-6-fluorophenyl)-3-(furan-2-yl)-8-meth...)
Affinity DataIC50:  3.00E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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