TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Inhibition of rat Nav1.2 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Siteone Therapeutics
Curated by ChEMBL
Siteone Therapeutics
Curated by ChEMBL
Affinity DataKd: 64nMAssay Description:Binding affinity to human recombinant Nav1.2 by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Siteone Therapeutics
Curated by ChEMBL
Siteone Therapeutics
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to human recombinant Nav1.2 by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Siteone Therapeutics
Curated by ChEMBL
Siteone Therapeutics
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Inhibition of full length human Nav1.2 expressed in HEK293 cells at -60 mV holding potential by manual patch clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 5.30nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 500nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 55nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair