TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.0160nMAssay Description:Binding affinity to Src (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Competitive inhibition of C-terminal His-tagged full length human SRC expressed in insect cells preincubated for 20 mins using poly[Glu,Tyr]4:1 as su...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 7.22nMAssay Description:Inhibition of Src by luminescence based kinase assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition of recombinant SRC (unknown origin) using polyE4Y as substrate by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Irreversible inhibition of wild type c-Src (unknown origin) assessed as inhibition constant by fluorimetric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 28.1nMAssay Description:Inhibition of Src by luminescence based kinase assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Inhibition of SrcChecked by AuthorMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Irreversible inhibition of wild type c-Src (unknown origin) assessed as inhibition constant by fluorimetric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair