Compile Data Set for Download or QSAR
Report error Found 155 Enz. Inhib. hit(s) with all data for entry = 2232
TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358552(US10214544, Example 52)
Affinity DataEC50:  0.410nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358797(US10214544, Example 110)
Affinity DataEC50:  0.520nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358233(US10214544, Example 17)
Affinity DataEC50:  0.550nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358799(US10214544, Example 112)
Affinity DataEC50:  0.550nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358566(US10214544, Example 58)
Affinity DataEC50:  0.740nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358408(US10214544, Example 26)
Affinity DataEC50:  0.75nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358548(US10214544, Example 49)
Affinity DataEC50:  0.850nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358409(US10214544, Example 27)
Affinity DataEC50:  0.870nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358234(US10214544, Example 18)
Affinity DataEC50:  0.910nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358769(US10214544, Example 74)
Affinity DataEC50:  0.950nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358838(US10214544, Example 153)
Affinity DataEC50:  0.990nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358488(US10214544, Example 35)
Affinity DataEC50:  1nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358160(US10214544, Example 2 | 4-Fluoro-N-(3-(((6-methoxy...)
Affinity DataEC50:  1nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358765(US10214544, Example 70)
Affinity DataEC50:  1nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358760(US10214544, Example 65)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358411(US10214544, Example 29)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358523(US10214544, Example 46)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358156(US10214544, Example 1 | N-(3-(((6-methoxy-2-(2-met...)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358784(US10214544, Example 90)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358265(US10214544, Example 22)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358561(US10214544, Example 55)
Affinity DataEC50:  1.10nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358487(US10214544, Example 34)
Affinity DataEC50:  1.20nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358473(US10214544, Example 31)
Affinity DataEC50:  1.30nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358837(US10214544, Example 152)
Affinity DataEC50:  1.30nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358827(US10214544, Example 142)
Affinity DataEC50:  1.30nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358183(US10214544, Example 5 | 4-Chloro-N-(3-(((6-methoxy...)
Affinity DataEC50:  1.30nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358759(US10214544, Example 64)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358222(US10214544, Example 16)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358220(US10214544, Example 14)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358758(US10214544, Example 63)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358259(US10214544, Example 20)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358280(US10214544, Example 24)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358504(US10214544, Example 40)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358187(US10214544, Example 6 | N-(3-(((6-methoxy-2-(2-met...)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358508(US10214544, Example 41)
Affinity DataEC50:  1.40nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358795(US10214544, Example 106)
Affinity DataEC50:  1.5nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358825(US10214544, Example 140)
Affinity DataEC50:  1.5nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358260(US10214544, Example 21)
Affinity DataEC50:  1.5nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358846(US10214544, Example 161)
Affinity DataEC50:  1.5nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358202(US10214544, Example 12)
Affinity DataEC50:  1.5nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358582(US10214544, Example 61)
Affinity DataEC50:  1.5nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358474(US10214544, Example 32)
Affinity DataEC50:  1.60nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358844(US10214544, Example 159)
Affinity DataEC50:  1.60nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358193(US10214544, Example 8)
Affinity DataEC50:  1.60nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358832(US10214544, Example 147)
Affinity DataEC50:  1.60nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358517(US10214544, Example 43)
Affinity DataEC50:  1.60nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358221(US10214544, Example 15)
Affinity DataEC50:  1.70nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358841(US10214544, Example 156)
Affinity DataEC50:  1.70nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358198(US10214544, Example 11)
Affinity DataEC50:  1.70nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358343(US10214544, Example 25)
Affinity DataEC50:  1.70nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

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