Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 12682
TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719141BDBM719141(N-((5-(2-fluorophenyl)-1-((4-fluorophenyl)sulfonyl...)
Affinity DataIC50: 25nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719140BDBM719140(N-((1-((4-chlorophenyl)sulfonyl)-5-(2-fluorophenyl...)
Affinity DataIC50: 26nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719139BDBM719139( N-((1-((4-bromophenyl)sulfonyl)-5-(2-fluorophenyl...)
Affinity DataIC50: 36nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719148BDBM719148(N-((4-methoxy-1-(pyridin-3-ylsulfonyl)-5-(2,4,6-tr...)
Affinity DataIC50: 38nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719135BDBM719135(N-((5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H...)
Affinity DataIC50: 42nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719137BDBM719137(N-((5-(2-fluorophenyl)-1-((4-methoxyphenyl)sulfony...)
Affinity DataIC50: 48nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719142BDBM719142(N-((5-(2-fluorophenyl)-1-((4-(trifluoromethoxy)phe...)
Affinity DataIC50: 51nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719143BDBM719143(N-((1-((4-chlorophenyl)sulfonyl)-5-(3-fluorophenyl...)
Affinity DataIC50: 60nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719149BDBM719149(N-((4-methoxy-1-((6-methoxypyridin-3-yl)sulfonyl)-...)
Affinity DataIC50: 64nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719136BDBM719136(N-((5-(2-fluorophenyl)-1-tosyl-1H-pyrrol-3-yl)meth...)
Affinity DataIC50: 68nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719144BDBM719144(N-((5-(3-fluorophenyl)-1-((4-methoxyphenyl)sulfony...)
Affinity DataIC50: 76nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719145BDBM719145(N-((5-(2,4-difluorophenyl)-1-tosyl-1H-pyrrol-3-yl)...)
Affinity DataIC50: 82nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719146BDBM719146(N-((5-(2,4-difluorophenyl)-1-((4-methoxyphenyl)sul...)
Affinity DataIC50: 84nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719147BDBM719147(N-((5-(2,4-difluorophenyl)-4-methoxy-1-((6-methoxy...)
Affinity DataIC50: 88nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Human)
Hana Pharm

US Patent
LigandChemical structure of BindingDB Monomer ID 719138BDBM719138(4-((2-(2-fluorophenyl)-4-(((methyl-d3)amino)methyl...)
Affinity DataIC50: 90nMAssay Description:60 ul of enzyme reaction solution (a test compound at a given concentration, 3 g of gastric mucosal microsomes, 3 mM of MgSO4, 5 mM of KCl, 40 mM of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
US Patent