Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 12934
TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50559373BDBM50559373(CHEMBL4795265 | US20250162994, Example 12)
Affinity DataIC50: 3nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50559389BDBM50559389(CHEMBL4762346 | US20250162994, Example 13)
Affinity DataIC50: 4nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50621126BDBM50621126(CHEMBL5407312 | US20250162994, Example 11)
Affinity DataIC50: 4nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741642BDBM741642(US20250162994, Example 25)
Affinity DataIC50: 4nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741621BDBM741621(N-hydroxy-4-(3-(4-((((1S,2R)-2-(1-phenyl-1H-pyrazo...)
Affinity DataIC50: 5nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741633BDBM741633(US20250162994, Example 16)
Affinity DataIC50: 5nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741643BDBM741643(US20250162994, Example 26)
Affinity DataIC50: 5nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741636BDBM741636(US20250162994, Example 19)
Affinity DataIC50: 6nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741644BDBM741644(US20250162994, Example 27)
Affinity DataIC50: 6nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741624BDBM741624(N-hydroxy-4-(3-(4-((((1R,2S)-2-(4-(pyrimidin-5-yl)...)
Affinity DataIC50: 6nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741641BDBM741641(US20250162994, Example 24)
Affinity DataIC50: 6nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50559388BDBM50559388(CHEMBL4749146 | US20250162994, Example 14)
Affinity DataIC50: 6nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741625BDBM741625(N-hydroxy-4-(3-(4-((((1S,2R)-2-(4-(pyrimidin-5-yl)...)
Affinity DataIC50: 8nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741620BDBM741620(N-hydroxy-4-(3-(4-((((1R,2S)-2-(1-phenyl-1H-pyrazo...)
Affinity DataIC50: 9nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741632BDBM741632(N-(2-aminophenyl)-4-(3-(4-((((1R,2S)-2-(4-fluoroph...)
Affinity DataIC50: 9nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741640BDBM741640(US20250162994, Example 23)
Affinity DataIC50: 10nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741467BDBM741467(N-hydroxy-4-((4-((((1R,2S)-2-phenylcyclopropyl)ami...)
Affinity DataIC50: 12nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741637BDBM741637(US20250162994, Example 20)
Affinity DataIC50: 20nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741647BDBM741647(US20250162994, Example 30)
Affinity DataIC50: 27nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741645BDBM741645(US20250162994, Example 28)
Affinity DataIC50: 29nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50559389BDBM50559389(CHEMBL4762346 | US20250162994, Example 13)
Affinity DataIC50: 31nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741622BDBM741622(4-((E)-3-(3-((((1R,2S)-2-(4-fluorophenyl)cycloprop...)
Affinity DataIC50: 31nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50621126BDBM50621126(CHEMBL5407312 | US20250162994, Example 11)
Affinity DataIC50: 31nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50559373BDBM50559373(CHEMBL4795265 | US20250162994, Example 12)
Affinity DataIC50: 54nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741467BDBM741467(N-hydroxy-4-((4-((((1R,2S)-2-phenylcyclopropyl)ami...)
Affinity DataIC50: 55nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741638BDBM741638(US20250162994, Example 21)
Affinity DataIC50: 69nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 50559388BDBM50559388(CHEMBL4749146 | US20250162994, Example 14)
Affinity DataIC50: 69nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741621BDBM741621(N-hydroxy-4-(3-(4-((((1S,2R)-2-(1-phenyl-1H-pyrazo...)
Affinity DataIC50: 72nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741622BDBM741622(4-((E)-3-(3-((((1R,2S)-2-(4-fluorophenyl)cycloprop...)
Affinity DataIC50: 84nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741620BDBM741620(N-hydroxy-4-(3-(4-((((1R,2S)-2-(1-phenyl-1H-pyrazo...)
Affinity DataIC50: 88nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741634BDBM741634(US20250162994, Example 17)
Affinity DataIC50: 101nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741627BDBM741627(N-hydroxy-4-(3-(4-((((1S,2R)-2-(1,3,3-trimethyl-2-...)
Affinity DataIC50: 135nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741635BDBM741635(US20250162994, Example 18)
Affinity DataIC50: 139nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741623BDBM741623(4-((E)-3-(3-((((1S,2R)-2-(4-fluorophenyl)cycloprop...)
Affinity DataIC50: 144nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741623BDBM741623(4-((E)-3-(3-((((1S,2R)-2-(4-fluorophenyl)cycloprop...)
Affinity DataIC50: 147nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741624BDBM741624(N-hydroxy-4-(3-(4-((((1R,2S)-2-(4-(pyrimidin-5-yl)...)
Affinity DataIC50: 151nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741625BDBM741625(N-hydroxy-4-(3-(4-((((1S,2R)-2-(4-(pyrimidin-5-yl)...)
Affinity DataIC50: 159nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741619BDBM741619(N-hydroxy-4-((4-((((1S,2R)-2-phenylcyclopropyl)ami...)
Affinity DataIC50: 178nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 1(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741647BDBM741647(US20250162994, Example 30)
Affinity DataIC50: 181nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741626BDBM741626(N-hydroxy-4-(3-(4-((((1R,2S)-2-(1,3,3-trimethyl-2-...)
Affinity DataIC50: 192nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 1(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741640BDBM741640(US20250162994, Example 23)
Affinity DataIC50: 262nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 1(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741633BDBM741633(US20250162994, Example 16)
Affinity DataIC50: 295nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741626BDBM741626(N-hydroxy-4-(3-(4-((((1R,2S)-2-(1,3,3-trimethyl-2-...)
Affinity DataIC50: 403nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741646BDBM741646(US20250162994, Example 29)
Affinity DataIC50: 671nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741639BDBM741639(US20250162994, Example 22)
Affinity DataIC50: 854nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 1(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741467BDBM741467(N-hydroxy-4-((4-((((1R,2S)-2-phenylcyclopropyl)ami...)
Affinity DataIC50: 923nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 1(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741634BDBM741634(US20250162994, Example 17)
Affinity DataIC50: 1.04E+3nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741627BDBM741627(N-hydroxy-4-(3-(4-((((1S,2R)-2-(1,3,3-trimethyl-2-...)
Affinity DataIC50: 1.21E+3nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741619BDBM741619(N-hydroxy-4-((4-((((1S,2R)-2-phenylcyclopropyl)ami...)
Affinity DataIC50: 1.34E+3nMAssay Description:LSD1 enzyme was produced in house. Tranylcypromine (TCP), LSD1 inhibitor was procured from Selleckchem. LSD1 enzyme, TCP and Biotinylated peptide sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetHistone deacetylase 1(Human)
Jubilant Epicore

US Patent
LigandChemical structure of BindingDB Monomer ID 741619BDBM741619(N-hydroxy-4-((4-((((1S,2R)-2-phenylcyclopropyl)ami...)
Affinity DataIC50: 1.55E+3nMAssay Description:Histone deacetylase assay was done as per manufacturer's instructions. Briefly, assay buffer, 200 uM HDAC substrate (fluorogenic HDAC acetylated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

Displayed 1 to 50 (of 57 total ) | Next | Last >>
Jump to: