Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 13332
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Pantherics Incorperated

US Patent
LigandChemical structure of BindingDB Monomer ID 781591BDBM781591(US20250319096, Compound PI531)
Affinity DataIC50: 31nMAssay Description:Rat brain membranes were prepared from frozen tissue that was thawed on ice and homogenized on ice in 10 volumes of cold lysis buffer (50 mM Tris HCl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/5/2026
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Pantherics Incorperated

US Patent
LigandChemical structure of BindingDB Monomer ID 781592BDBM781592(US20250319096, Compound PI352)
Affinity DataIC50: 38nMAssay Description:Rat brain membranes were prepared from frozen tissue that was thawed on ice and homogenized on ice in 10 volumes of cold lysis buffer (50 mM Tris HCl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/5/2026
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Pantherics Incorperated

US Patent
LigandChemical structure of BindingDB Monomer ID 781590BDBM781590(US20250319096, Compound PI350)
Affinity DataIC50: 58nMAssay Description:Rat brain membranes were prepared from frozen tissue that was thawed on ice and homogenized on ice in 10 volumes of cold lysis buffer (50 mM Tris HCl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/5/2026
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Pantherics Incorperated

US Patent
LigandChemical structure of BindingDB Monomer ID 781589BDBM781589(US20250319096, Compound PI320)
Affinity DataIC50: 242nMAssay Description:Rat brain membranes were prepared from frozen tissue that was thawed on ice and homogenized on ice in 10 volumes of cold lysis buffer (50 mM Tris HCl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/5/2026
Entry Details
US Patent