Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
Report error
Found
22
Enz. Inhib. hit(s) with all data for entry = 13348
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782791
(6-(6-(((1S,3S)-3-((5-(2,2,2-trifluoroethoxyl)pyrim...)
Copy SMILES
Affinity Data
Kd: 0.800nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782795
(US20250326722, Example 132)
Copy SMILES
Affinity Data
Kd: 1.10nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782797
(6-(6-(((1S,3S)-3-((7-(trifluoromethyl)-[1,2,4]tria...)
Copy SMILES
Affinity Data
Kd: 1.20nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782794
(6-(6-(((1S,3S)-3-((7-methyl-[1,2,4]triazolo[1,5-a]...)
Copy SMILES
Affinity Data
Kd: 1.20nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782792
(6-(6-(((1S,3S)-3-((6-cyclopropyl-1,2,4-triazin-3-y...)
Copy SMILES
Affinity Data
Kd: 1.20nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782800
(2-(6-(((1S,3S)-3-((7-fluoro-[1,2,4]triazolo[1,5-a]...)
Copy SMILES
Affinity Data
Kd: 1.40nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782785
(6-(6-(((1S,3S)-3-((5-(difluoromethoxy)pyrimidin-2-...)
Copy SMILES
Affinity Data
Kd: 1.5nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782793
(6-(6-(((1S,3S)-3-((5-cyclopropylpyrimidin-2-yl)ami...)
Copy SMILES
Affinity Data
Kd: 1.80nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782790
(6-(6-(((1S,3S)-3-((5-(trifluoromethoxy)pyrimidin-2...)
Copy SMILES
Affinity Data
Kd: 2.20nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782783
(6'-(((1S,3S)-3-(pyrrolo[2,1-f][1,2,4]triazin-2-yla...)
Copy SMILES
Affinity Data
Kd: 2.40nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782799
(US20250326722, Example 146)
Copy SMILES
Affinity Data
Kd: 2.5nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782784
(6'-((3-(((1S,3S)-7-fluoro-[1,2,4]triazolo[1,5-a]py...)
Copy SMILES
Affinity Data
Kd: 2.60nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782803
(2-(6-(((1S,3S)-3-((7-fluoro-[1,2,4]triazolo[1,5-a]...)
Copy SMILES
Affinity Data
Kd: 2.60nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782787
(6'-(((1S,3S)-3-((7-chloro-[1,2,4]triazolo[1,5-a]py...)
Copy SMILES
Affinity Data
Kd: 2.70nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782801
(6-(6-(((1S,3S)-3-((7-fluoro-[1,2,4]triazolo[1,5-a]...)
Copy SMILES
Affinity Data
Kd: 2.80nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782786
(US20250326722, Example 93)
Copy SMILES
Affinity Data
Kd: 2.90nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782804
(2-(6-(((1S,3S)-3-((7-fluoro-[1,2,4]triazolo[1,5-a]...)
Copy SMILES
Affinity Data
Kd: 3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782789
(2-(6-(((1S,3S)-3-((5-(difluoromethoxy)pyrimidin-2-...)
Copy SMILES
Affinity Data
Kd: 3.10nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782798
(US20250326722, Example 145)
Copy SMILES
Affinity Data
Kd: 3.20nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782788
(6'-(((1S,3S)-3-((7-(trifluoromethyl)-[1,2,4]triazo...)
Copy SMILES
Affinity Data
Kd: 4.20nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782802
(6-Methyl-2-(6-(((1S,3S)-3-((7-(trifluoromethyl)-[1...)
Copy SMILES
Affinity Data
Kd: 4.80nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
Target
Proprotein convertase subtilisin/kexin type 9
(Human)
Shanghai Hansoh Biomedical Co.
US Patent
Ligand
BDBM782796
(6'-(((1S,3S)-3-((7-cyclopropyl-[1,2,4]triazolo[1,5...)
Copy SMILES
Affinity Data
Kd: 4.90nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
2/11/2026
Entry Details
US Patent
Copy reaction URL
BDBM782794
