Compile Data Set for Download or QSAR
Report error Found 1030 Enz. Inhib. hit(s) with all data for entry = 5902
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99618BDBM99618(US8501936, 119)
Affinity DataIC50: 0.270nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99529BDBM99529(CHEMBL2062802 | US8501936, 27)
Affinity DataIC50: 0.400nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99683BDBM99683(US8501936, 184)
Affinity DataIC50: 0.410nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99689BDBM99689(US8501936, 190)
Affinity DataIC50: 0.460nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99710BDBM99710(US8501936, 212)
Affinity DataIC50: 0.5nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99620BDBM99620(US8501936, 121)
Affinity DataIC50: 0.550nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99690BDBM99690(US8501936, 191)
Affinity DataIC50: 0.550nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99548BDBM99548(US8501936, 46)
Affinity DataIC50: 0.600nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99520BDBM99520(US8501936, 18)
Affinity DataIC50: 0.600nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99565BDBM99565(US8501936, 63)
Affinity DataIC50: 0.600nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99564BDBM99564(US8501936, 62)
Affinity DataIC50: 0.600nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99682BDBM99682(US8501936, 183)
Affinity DataIC50: 0.650nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99614BDBM99614(US8501936, 115)
Affinity DataIC50: 0.660nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99619BDBM99619(CHEMBL2062807 | US8501936, 120)
Affinity DataIC50: 0.670nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99550BDBM99550(US8501936, 48)
Affinity DataIC50: 0.700nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99516BDBM99516(US8501936, 12)
Affinity DataIC50: 0.700nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99563BDBM99563(CHEMBL2062809 | US8501936, 61)
Affinity DataIC50: 0.700nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99711BDBM99711(US8501936, 213)
Affinity DataIC50: 0.710nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99667BDBM99667(US8501936, 168)
Affinity DataIC50: 0.730nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99641BDBM99641(US8501936, 142)
Affinity DataIC50: 0.75nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99613BDBM99613(US8501936, 114)
Affinity DataIC50: 0.75nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99573BDBM99573(US8501936, 71)
Affinity DataIC50: 0.800nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 50389186BDBM50389186(CHEMBL2062803 | US8501936, 4)
Affinity DataIC50: 0.900nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99616BDBM99616(US8501936, 117)
Affinity DataIC50: 0.950nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99680BDBM99680(US8501936, 181)
Affinity DataIC50: 0.970nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99521BDBM99521(CHEMBL2062799 | US8501936, 19)
Affinity DataIC50: 1nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99536BDBM99536(US8501936, 34)
Affinity DataIC50: 1nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99542BDBM99542(CHEMBL2062798 | US8501936, 40)
Affinity DataIC50: 1nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99514BDBM99514(US8501936, 10)
Affinity DataIC50: 1nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99596BDBM99596(US8501936, 95)
Affinity DataIC50: 1nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99767BDBM99767(US8501936, 283)
Affinity DataIC50: 1.06nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99552BDBM99552(US8501936, 50)
Affinity DataIC50: 1.10nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99572BDBM99572(US8501936, 70)
Affinity DataIC50: 1.10nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99586BDBM99586(US8501936, 85)
Affinity DataIC50: 1.10nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99642BDBM99642(US8501936, 143)
Affinity DataIC50: 1.13nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99555BDBM99555(CHEMBL2062810 | US8501936, 53)
Affinity DataIC50: 1.30nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99537BDBM99537(CHEMBL2062804 | US8501936, 35)
Affinity DataIC50: 1.30nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99576BDBM99576(US8501936, 75)
Affinity DataIC50: 1.30nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99611BDBM99611(CHEMBL2062801 | US8501936, 112)
Affinity DataIC50: 1.30nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99528BDBM99528(US8501936, 26)
Affinity DataIC50: 1.30nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99685BDBM99685(US8501936, 186)
Affinity DataIC50: 1.35nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99594BDBM99594(US8501936, 93)
Affinity DataIC50: 1.40nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99617BDBM99617(US8501936, 118)
Affinity DataIC50: 1.43nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99687BDBM99687(US8501936, 188)
Affinity DataIC50: 1.43nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99560BDBM99560(CHEMBL2062529 | US8501936, 58)
Affinity DataIC50: 1.5nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99550BDBM99550(US8501936, 48)
Affinity DataIC50: 1.5nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99644BDBM99644(US8501936, 145)
Affinity DataIC50: 1.55nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99892BDBM99892(US8501936, 411)
Affinity DataIC50: 1.62nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99702BDBM99702(US8501936, 204)
Affinity DataIC50: 1.63nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Cephalon

US Patent
LigandChemical structure of BindingDB Monomer ID 99556BDBM99556(US8501936, 54)
Affinity DataIC50: 1.70nMAssay Description:The ability of compounds to inhibit the kinase activity of baculovirus-expressed human FAK and JAK kinase using the time-resolved fluorescence (TRF) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

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